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Anzahl der Publikationen: 13
Zeitschriftenartikel
Hluchy, Milan; Gajduskova, Pavla; Ruiz de los Mozos, Igor; Rajecky, Michal; Kluge, Michael; Berger, Benedict-Tilman; Slaba, Zuzana; Potesil, David; Weiss, Elena; Ule, Jernej; Zdrahal, Zbynek; Knapp, Stefan; Paruch, Kamil; Friedel, Caroline C. und Blazek, Dalibor
(2022):
CDK11 regulates pre-mRNA splicing by phosphorylation ofSF3B1.
In: Nature, Bd. 609, Nr. 7928: S. 829-834
Arifi, Silvia; Zaienne, Daniel; Heering, Jan; Wein, Thomas; Zhubi, Rezart; Chaikuad, Apirat; Knapp, Stefan; Marschner, Julian A. und Merk, Daniel
(2022):
Fragment-based discovery of orphan nuclear receptor Nur77/NGFI-B ligands.
In: Bioorganic Chemistry, Bd. 129, 106164
Faudone, Giuseppe; Zhubi, Rezart; Celik, Fatih; Knapp, Stefan; Chaikuad, Apirat; Heering, Jan und Merk, Daniel
(2022):
Design of a Potent TLX Agonist by Rational Fragment Fusion.
In: Journal of Medicinal Chemistry, Bd. 65, Nr. 3: S. 2288-2296
Faudone, Giuseppe; Kilu, Whitney; Ni, Xiaomin; Chaikuad, Apirat; Sreeramulu, Sridhar; Heitel, Pascal; Schwalbe, Harald; Knapp, Stefan; Schubert-Zsilavecz, Manfred; Heering, Jan und Merk, Daniel
(2021):
The Transcriptional Repressor Orphan Nuclear Receptor TLX Is Responsive to Xanthines.
In: ACS Pharmacology & Translational Science, Bd. 4, Nr. 6: S. 1794-1807
Krishnathas, G. Melissa; Strödke, Benjamin; Mittmann, Laura; Zech, Thomas; Berger, Lena M.; Reichel, Christoph A.; Rösser, Silvia; Schmid, Tobias; Knapp, Stefan; Müller, Susanne; Bracher, Franz; Fürst, Robert und Bischoff-Kont, Iris
(2021):
C81-evoked inhibition of the TNFR1-NF kappa B pathway during inflammatory processes for stabilization of the impaired vascular endothelial barrier for leukocytes.
In: Faseb Journal, Bd. 35, Nr. 6, e21656
Mueller, Susanne; Ackloo, Suzanne; Al Chawaf, Arij; Al-Lazikani, Bissan; Antolin, Albert; Baell, Jonathan B.; Beck, Hartmut; Beedie, Shaunna; Betz, Ulrich A. K.; Bezerra, Gustavo Arruda; Brennan, Paul E.; Brown, David; Brown, Peter J.; Bullock, Alex N.; Carter, Adrian J.; Chaikuad, Apirat; Chaineau, Mathilde; Ciulli, Alessio; Collins, Ian; Dreher, Jan; Drewry, David; Edfeldt, Kristina; Edwards, Aled M.; Egner, Ursula; Frye, Stephen V.; Fuchs, Stephen M.; Hall, Matthew D.; Hartung, Ingo V.; Hillisch, Alexander; Hitchcock, Stephen H.; Homan, Evert; Kannan, Natarajan; Kiefer, James R.; Knapp, Stefan; Kostic, Milka; Kubicek, Stefan; Leach, Andrew R.; Lindemann, Sven; Marsden, Brian D.; Matsui, Hisanori; Meier, Jordan L.; Merk, Daniel; Michel, Maurice; Morgan, Maxwell R.; Mueller-Fahrnow, Anke; Owen, Dafydd R.; Perry, Benjamin G.; Rosenberg, Saul H.; Saikatendu, Kumar Singh; Schapira, Matthieu; Scholten, Cora; Sharma, Sujata; Simeonov, Anton; Sundstrom, Michael; Superti-Furga, Giulio; Todd, Matthew H.; Tredup, Claudia; Vedadi, Masoud; Delft, Frank von; Willson, Timothy M.; Winter, Georg E.; Workman, Paul und Arrowsmith, Cheryl H.
(2021):
Target 2035-update on the quest for a probe for every protein.
In: Rsc Medicinal Chemistry, Bd. 13, Nr. 1: S. 13-21
Reynders, Martin; Chaikuad, Apirat; Berger, Benedict-Tilman; Bauer, Katharina; Koch, Pierre; Laufer, Stefan; Knapp, Stefan und Trauner, Dirk
(2021):
Controlling the Covalent Reactivity of a Kinase Inhibitor with Light.
In: Angewandte Chemie-International Edition, Bd. 60, Nr. 37: S. 20178-20183
Schroeder, Martin; Bullock, Alex N.; Fedorov, Oleg; Bracher, Franz; Chaikuad, Apirat und Knapp, Stefan
(2020):
DFG-1 Residue Controls Inhibitor Binding Mode and Affinity, Providing a Basis for Rational Design of Kinase Inhibitor Selectivity.
In: Journal of Medicinal Chemistry, Bd. 63, Nr. 18: S. 10224-10234
Wurzlbauer, Anne; Rueben, Katharina; Guerdal, Ece; Chaikuad, Apirat; Knapp, Stefan; Sippl, Wolfgang; Becker, Walter und Bracher, Franz
(2020):
How to Separate Kinase Inhibition from Undesired Monoamine Oxidase A Inhibition-The Development of the DYRK1A Inhibitor AnnH75 from the Alkaloid Harmine.
In: Molecules, Bd. 25, Nr. 24, 5962
Tuppi, Marcel; Kehrloesser, Sebastian; Coutandin, Daniel W.; Rossi, Valerio; Luh, Laura M.; Strubel, Alexander; Hoette, Katharina; Hoffmeister, Meike; Schaefer, Birgit; De Oliveira, Tiago; Greten, Florian; Stelzer, Ernst H. K.; Knapp, Stefan; Felici, Massimo de; Behrends, Christian; Klinger, Francesca Gioia und Doetsch, Volker
(2018):
Oocyte DNA damage quality control requires consecutive interplay of CHK2 and CK1 to activate p63.
In: Nature Structural & Molecular Biology, Bd. 25, Nr. 3: S. 261-269
Moustakim, Moses; Riedel, Kerstin; Schuller, Marion; Gehring, Andre P.; Monteiro, Octovia P.; Martin, Sarah P.; Fedorov, Oleg; Heer, Jag; Dixon, Darren J.; Elkins, Jonathan M.; Knapp, Stefan; Bracher, Franz und Brennan, Paul E.
(2018):
Discovery of a novel allosteric inhibitor scaffold for polyadenosine-diphosphate-ribose polymerase 14 (PARP14) macrodomain 2.
In: Bioorganic & Medicinal Chemistry, Bd. 26, Nr. 11: S. 2965-2972
Schuller, Marion; Riede, Kerstin; Gibbs-Seymour, Ian; Uth, Kristin; Sieg, Christian; Gehring, Andre P.; Ahel, Ivan; Bracher, Franz; Kessler, Benedikt M.; Elkins, Jonathan M. und Knapp, Stefan
(2017):
Discovery of a Selective Allosteric Inhibitor Targeting Macrodomain 2 of Polyadenosine-Diphosphate-Ribose Polymerase 14.
In: ACS Chemical Biology, Bd. 12, Nr. 11: S. 2866-2874
Popp, Tobias A.; Tallant, Cynthia; Rogers, Catherine; Fedorov, Oleg; Brennan, Paul E.; Müller, Susanne; Knapp, Stefan und Bracher, Franz
(2016):
Development of Selective CBP/P300 Benzoxazepine Bromodomain Inhibitors.
In: Journal of Medicinal Chemistry, Bd. 59, Nr. 19: S. 8889-8912